AUTHOR=De Surya K. TITLE=Leniolisib: a novel treatment for activated phosphoinositide-3 kinase delta syndrome JOURNAL=Frontiers in Pharmacology VOLUME=15 YEAR=2024 URL=https://www.frontiersin.org/journals/pharmacology/articles/10.3389/fphar.2024.1337436 DOI=10.3389/fphar.2024.1337436 ISSN=1663-9812 ABSTRACT=Graphical Abstract

IC50 = 11 nM (PI3Kδ); 244 nM (PI3Kα); 424 nM (PI3Kβ), 2,230 nM (PI3Kγ).